中文名 | 凝血酶受体激活肽6 |
英文名 | TRAP-6 |
别名 | TRAP-6游离态 凝血酶受体激活肽6 化合物TRAP-6(2TFA) |
英文别名 | TRAP-6 TRAP-6(2TFA) SER-PHE-LEU-LEU-ARG-ASN H-SER-PHE-LEU-LEU-ARG-ASN-OH TRAP-6SER-PHE-LEU-LEU-ARG-ASN THROMBIN RECEPTOR (42-47), HUMAN L-Asparagine,L-seryl-L-phenylalanyl-L-leucyl-L-leucyl-L-arginyl- |
CAS | 141136-83-6 |
化学式 | C34H56N10O9 |
分子量 | 748.87 |
水溶性 | Soluble in water at 1mg/ml |
溶解度 | TFA 0.1%: 可溶性 |
存储条件 | -20°C |
物化性质 | 溶解度:TFA 0.1%: soluble 储存条件:?20℃ WGK Germany:3 |
体外研究 | TRAP-6 (0.01-10 μM) triggers calcium mobilization in Xenopus oocytes heterologously expressing PAR1. TRAP-6 (0.01-10 μM; 30 min) activates human platelets. TRAP-6 (100 μM) does not cause the platelets of rabbits or rats to change shape, aggregate, release granule contents, or form thromboxane. |
体内研究 | TRAP (1 mg/kg; i.v.) produces a biphasic response in blood pressure in inactin-anesthetized rats. |
WGK Germany | 3 |
1mg | 5mg | 10mg | |
---|---|---|---|
1 mM | 1.335 ml | 6.677 ml | 13.353 ml |
5 mM | 0.267 ml | 1.335 ml | 2.671 ml |
10 mM | 0.134 ml | 0.668 ml | 1.335 ml |
5 mM | 0.027 ml | 0.134 ml | 0.267 ml |