GALUNISERTIB
LY 2157299
CAS: 700874-72-2
Molecular Formula: C22H19N5O
GALUNISERTIB - Names and Identifiers
GALUNISERTIB - Physico-chemical Properties
| Molecular Formula | C22H19N5O |
| Molar Mass | 369.42 |
| Density | 1.40 |
| Melting Point | 241-242°C |
| Boling Point | 619.0±55.0 °C(Predicted) |
| Flash Point | 328.162℃ |
| Solubility | DMSO 74 mg/mL (200.31 mM); Water <1 mg/mL (<1 mM);Ethanol <1 mg/mL (<1 mM) |
| Appearance | Form solid, color White |
| Storage Condition | -20°C |
| Stability | Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month. |
| Physical and Chemical Properties | Bioactive Galunisertib (LY2157299) is a potent TGF β receptor I (TβRI) inhibitor with an IC50 of 56 nM in cell-free assays. Phase 2/3. |
| Use | The LY2157299 of use is TGF-βI receptor kinase inhibitor. LY2157299 has been used to enhance chemotherapy for triple negative breast cancer (TNBC). |
GALUNISERTIB - Risk and Safety
| Hazard Symbols | T - Toxic |
| Risk Codes | 25 - Toxic if swallowed |
| Safety Description | 45 - In case of accident or if you feel unwell, seek medical advice immediately (show the label whenever possible.) |
| HS Code | 29334900 |
GALUNISERTIB - Upstream Downstream Industry
GALUNISERTIB - Introduction
LY2157299 is a potent TGF β receptor I (TβRI) inhibitor with an IC50 of 56 nM. Phase 2/3.
Last Update：2022-10-16 17:30:55
GALUNISERTIB - Nature
| Solubility | Soluble in DMSO (up to 25 mg/ml) |
Last Update：2024-04-10 22:29:15
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View History
Raw Materials for GALUNISERTIB
6-Quinolinecarboxylic acid, 4-[5,6-dihydro-2-(6-Methyl-2-pyridinyl)-4H-pyrrolo[1,2-b]pyrazol-3-yl]-, Methyl ester
4-(2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)quinoline-6-carbonitrile
4-(2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)quinoline-6-carbonitrile