Molecular Formula | C28H35N5O4 |
Molar Mass | 505.61 |
Density | 1.25 |
pKa | 15?+-.0.46(Predicted) |
uses | captorelin is a ghrelin agonist useful in the treatment of insulin resistance in mammals. |
biological activity | Capromorelin Tartrate (CP 424391-18) is a growth hormone secretagogue (GHS) class of drugs, it is an agonist of ghrelin receptor and can be used as a new type of appetite stimulating therapy in dogs, with a Ki value of 7 nM for hGHS-R1a and an EC50 value of 3 nM for rat pituitary cells. |
Target | Value |
rat pituicyte (Cell-free assay) | 3 nM(EC50) |
hGHS-R1a (Cell-free assay) | 7 nM(Ki) |