Molecular Formula | C11H13NOS |
Molar Mass | 207.29 |
Solubility | DMSO: ≥ 28 mg/mL |
Storage Condition | Sealed in dry,Store in freezer, under -20°C |
1mg | 5mg | 10mg | |
---|---|---|---|
1 mM | 4.824 ml | 24.121 ml | 48.241 ml |
5 mM | 0.965 ml | 4.824 ml | 9.648 ml |
10 mM | 0.482 ml | 2.412 ml | 4.824 ml |
5 mM | 0.096 ml | 0.482 ml | 0.965 ml |
Biological activity | K-Ras-IN-1 (MDK-3017) can inhibit K-Ras by combining K-Ras in the hydrophobic pocket occupied by Tyr-71 in the apo-Ras crystal structure. |
target | TargetValue K-ras () |
Target | Value |