Molecular Formula | C9H9BrN2O3 |
Molar Mass | 273.08 |
Density | 1.711 |
Melting Point | 144°C(lit.) |
Solubility | DMSO: ≥5mg/mL |
Appearance | White solid |
Color | white to tan |
Storage Condition | 2-8°C |
MDL | MFCD00116442 |
In vitro study | Bikinin directly targets BIN2 of Arabidopsis GSK-3s and activates brassinosteroid-dependent gene expression. Bikinin also inhibits RD26 expression, and inhibits the induction of GUS activity by 150 mM NaCl in the RD26pro:GUS line. |
In vivo study | Bikinin strongly inhibits abscisic acid signaling outputs, and inhibits T180 phosphorylation of SnRK2.3 and its kinase activity in vivo. |
Hazard Symbols | Xn - Harmful |
Risk Codes | R22 - Harmful if swallowed R36 - Irritating to the eyes |
Safety Description | 26 - In case of contact with eyes, rinse immediately with plenty of water and seek medical advice. |
WGK Germany | 3 |
Reference Show more | 1. [IF=5.923] Jingjue Zeng et al."Functional Characterization of VvSK Gene Family in Grapevine Revealing Their Role in Berry Ripening."Int J Mol Sci. 2020 Jan;21(12):4336 |
1mg | 5mg | 10mg | |
---|---|---|---|
1 mM | 3.662 ml | 18.309 ml | 36.618 ml |
5 mM | 0.732 ml | 3.662 ml | 7.324 ml |
10 mM | 0.366 ml | 1.831 ml | 3.662 ml |
5 mM | 0.073 ml | 0.366 ml | 0.732 ml |
biological activity | Bikinin is an ATP competitive Arabidopsis GSK-3 inhibitor, which acts as a potent activator of brassinosteroid (BR) signal. |
in vitro study | Bikinin directly targets BIN2 of Arabidopsis GSK-3s and activates brassinosteroid-dependent gene expression. Bikinin also inhibits RD26 expression, and inhibits the induction of GUS activity by 150 mM NaCl in the RD26pro:GUS line. |
in vivo study | Bikinin strongly inhibits abscisic acid signaling outputs, and inhibits T180 phosphorylation of SnRK2.3 and its kinase activity in vivo. |
target | GSK-3 |