Cetrorelix diacetate MedChemExpress (MCE)

Product Name	Cetrorelix acetate
Synonyms	Cetrelix Acetate NS-75A diacetate SB-075 diacetate Cetrorelix acetate Cetrorenlin Acetate Cetrorelix Diacetate N-Acetyl-3-(2-naphthalenyl)-D-alanyl-4-chloro-D-phenylalanyl-3-(3-pyridinyl)-D-alanyl-L-seryl-L-tyrosyl-N5-(aminocarbonyl)-D-ornithyl-L-leucyl-L-arginyl-L-prolyl-D-alaninamide diacetate
CAS	130143-01-0
EINECS
Chemical Formula	C70H92N17O14
Molecular Weight	1551.16
inchi
Package	Inquiry
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Descriptions	Cetrorelix diacetate Cetrorelix diacetate MedChemExpress (MCE) HY-P0009B 130143-01-0 SB-75 diacetate Please store the product under the recommended conditions in the Certificate of Analysis. Room temperature in continental US Descriptions Cetrorelix diacetate Cetrorelix diacetate MedChemExpress (MCE) HY-P0009B 130143-01-0 SB-75 diacetate Please store the product under the recommended conditions in the Certificate of Analysis. Room temperature in continental US may vary elsewhere. Cetrorelix diacetate (SB-075 diacetate) is a potent gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM. Cetrorelix diacetate inhibits growth of ES-2 cell line at 1000 ng/ml. Cetrorelix diacetate has comparable antiproliferative effects as GnRH-I agonists indicating that the dichotomy of GnRH-I agonists and antagonists might not apply to the GnRH-I system in cancer cells[2]. IC50: 1.21 nM GnRH[1]. In Vitro Cetrorelix diacetate inhibits growth of ES-2 cell line at 1000 ng/ml. Cetrorelix diacetate has comparable antiproliferative effects as GnRH-I agonists indicating that the dichotomy of GnRH-I agonists and antagonists might not apply to the GnRH-I system in cancer cells[2]. MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only. 0 --> Cetrorelix diacetate Related Antibodies \| \| \| \| \| \| \| \| \| \| [1]. Beckers T et al. Characterization of gonadotropin-releasing hormone analogs based on a sensitive cellular luciferase reporter gene assay. Anal Biochem. 1997 Aug 15 251(1):17-23. [Content Brief] [2]. Gründker C et al. Role of gonadotropin-releasing hormone (GnRH) in ovarian cancer. Reprod Biol Endocrinol. 2003 Oct 7 1:65. [Content Brief]
Supplier Website	https://www.medchemexpress.com/cetrorelix-diacetate.html
Last Update	2025-05-21 16:50:25

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