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中文名 | 环丙基[4-[3-(1H-咪唑-5-基)丙氧基]苯基]甲酮盐酸盐 |
英文名 | Cyclopropyl[4-[3-(1H-imidazol-5-yl)propoxy]phenyl]methanone hydrochloride |
别名 | 环丙基[4-[3-(1H-咪唑-5-基)丙氧基]苯基]甲酮盐酸盐 |
CAS | 1049741-81-2 |
EINECS | |
化学式 | C16H19ClN2O2 |
分子量 | 306.78726 |
inchi | |
包装信息 | 5mg |
价格 | 1942 |
产品描述 | Ciproxifan belongs to a novel chemical series of histamine H3-receptor antagonists. In vitro, it behaved as a competitive antagonist at the H3 autoreceptor controlling 3H histamine release from synaptosomes and displayed similar Ki values (0.5-1.9 nM) at the H3 receptor controlling the electrically-induced contraction of guinea pig ileum or at the brain H3 receptor labeled with 125I-iodoproxyfan. Ciproxifan appears to be an orally bioavailable, extremely potent and selective H3-receptor antagonist whose vigilance- and attention-promoting effects are promising for therapeutic applications in aging disorders. |
更新日期 | 2023-12-05 15:37:59 |